Abstract
A central process contributing to the phenotype of aging is cellular senescence. We recently identified the FOXO4 - p53 axis as pivotal in maintaining the viability of senescent cells, and that senescent cells can be targeted selectively with the senolytic peptide FOXO4-DRI. Here, we solve the solution NMR structural models of the p53 transactivation domain in complex with the FOXO4 forkhead domain and in complex with FOXO4-DRI. Strikingly, we find that the disordered FOXO4-DRI binds to the disordered p53TAD2 and forms a transiently folded complex. In this complex, both, the FOXO4-derived region and the cationic cell permeability peptide contribute to the interaction. Furthermore, we show that p53 phosphorylation enhances the affinity for both FOXO4 and FOXO4-DRI. Summarizing we provide a detailed characterization of the interaction of p53 with FOXO4 and FOXO4-DRI which is the basis for development of p53 inhibitors to treat diseases linked to cellular senescence such as cancers.
| Original language | English |
|---|---|
| Article number | 5672 |
| Journal | Nature Communications |
| Volume | 16 |
| Issue number | 1 |
| DOIs | |
| Publication status | Published - 1 Jul 2025 |
Keywords
- Cell Cycle Proteins/metabolism
- Cellular Senescence
- Forkhead Transcription Factors/metabolism
- Humans
- Models, Molecular
- Phosphorylation
- Protein Binding
- Protein Domains
- Transcription Factors/metabolism
- Transcriptional Activation
- Tumor Suppressor Protein p53/metabolism
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